Ana sayfa | İletişim | English

Doç.Dr. Ş.Güniz Küçükgüzel'in resmi internet sitesi

 

BİLDİRİLER

 

Uluslararası Kongreler

1.

Kömürcü, Ş.G., M.Ülgen, S.Rollas ve S.Sezen . “The in-vitro hepatic oxidative microsomal metabolism of 4-aminobenzoic acid-p-fluorobenzalhydrazone” 53rd International Congress of Pharmaceutical Sciences, Tokyo-JAPAN, Abstract p.68, 6-10 September 1993.

2.

Kömürcü, Ş.G., S.Rollas, N.Yılmaz, T.Akkoç ve A.Çevikbaş . “Synthesis of  3-Methyl-[(2,4-dihydro-4-substituted-3H-1,2,4-triazole-3-thione-5-yl)phenylhydrazono]-5-isoxazolone and Evaluation of Their Antimicrobial Activities”, First International Meeting on Pharmacy & Pharmaceutical Sciences, İstanbul-TURKEY, J.Pharm.Uni.Mar. 10, supplement, p.168, 4-7 September 1994.

3.

Kömürcü, Ş.G., S.Rollas, T.Akkoç ve A.Çevikbaş. “Synthesis of  p-(acetylacetonylidene hydrazino)-[(substituted phenyl/pyridyl)methylene]benzoic acid hydrazide and Evaluation of Their Antimicrobial Activities”, First International Meeting on Pharmacy & Pharmaceutical Sciences, İstanbul-TURKEY, J.Pharm.Uni.Mar. 10, supplement, p.169, 4-7 September 1994.

4.

Kömürcü, Ş.G., İ.Küçükgüzel ve S.Rollas. “Synthesis,  Characterizations and Biological Evaluation of 3-Methyl-4-{4-[3-[(substituted benzyl)thio]-4-alkyl/aryl-4H-1,2,4-triazole-5-yl]phenylhydrazono}-5-isoxazolones”, 4th International Symposium on Pharmaceutical Sciences , Ankara-TURKEY, Abstract P-103, 27-30 June 1995.

5.

Küçükgüzel, İ., Ş.G.Kömürcü and S.Rollas. “Synthesis and Characterization of Some Novel 1,2,4-Triazoles as Potential Antimicrobial Agents”, 4th International Symposium on Pharmaceutical Sciences , Ankara-TURKEY, Abstract O-13, 27-30 June 1995.

6.

Küçükgüzel, İ., S.Rollas, Ş.G.Küçükgüzel and M.Kiraz .“Synthesis, Characterization and Antimycobacterial Activity of Some Thiourea Derivatives Obtained from 1,2,4-Triazoles”, XIVth International Symposium on Medicinal Chemistry , Maastricht-Netherlands , Abstract P-10.12, 8-12 September 1996 .

7.

Küçükgüzel, Ş.G., S.Rollas, İ.Küçükgüzel and M.Kiraz. “Synthesis and Antimycobacterial Activity of Some Coupling Products from 4-Aminobenzoic acid hydrazones”, XIVth International Symposium on Medicinal Chemistry , Maastricht-Netherlands , Abstract P-10.13, 8-12 September 1996 .

8.

Küçükgüzel, Ş.G., S.Rollas, H.Erdeniz, M.Kiraz . “Synthesis, Characterization and Antimicrobial Evaluation of Ethyl 2-arylhydrazono-3-oxobutyrates”,Drug Metabolism: Towards the Next Millennium, Chelsea, Abstract P-5, 26-28 August 1997.

9.

Küçükgüzel, Ş.G., S.Rollas, H.Erdeniz, M.Kiraz. “Synthesis, Characterization and Antimicrobial Evaluation of 4-arylhydrazono-2-pyrazoline-5-ones”, First International Symposium on Pharmaceutical Chemistry, Ankara-TURKEY, Abstract P-034, 24-26 September 1997.

10.

Küçükgüzel, Ş.G., İ.Küçükgüzel, M.Ülgen. “In vitro Microsomal Metabolism of N-(4-chlorobenzyl)-N’-benzoylhydrazine” , Second International Meeting on Pharmacy & Pharmaceutical Sciences, İstanbul-TURKEY, Abstract P 75, 6-9  September 1998.

11.

Küçükgüzel, İ., Ş.G.Küçükgüzel, S.Rollas, G.Ötük, O.Özdemir, T.Altuğ and İ.Bayrak. “Some Novel 1,2,4-Triazoles: Synthesis, Characterization and Evaluation of Antimicrobial and Anticonvulsant Activity”, Second International Meeting on Pharmacy & Pharmaceutical Sciences, İstanbul-TURKEY, Abstract P 74, 6-9 September 1998.

12.

Oruç, E.E., Ş.G. Küçükgüzel, S. Rollas. “Synthesis and Characterization of some novel hydrazones and thiosemicarbazides of 4-(4-methoxybenzoylamino)benzoyl hydrazine” 2nd  International Symposium on Pharmaceutical Chemistry, Ankara-TURKEY, Abstract P-04, 22-24 September 1999.

13.

Küçükgüzel, Ş.G., İ.Küçükgüzel, M.Ülgen. “Metabolic and Chemical Studies on N-(4-chlorobenzyl)-N’-benzoylhydrazine” 9th North American ISSX Meeting , Nashville, Tennessee-USA, P-223, 24-28 October 1999.

14.

Küçükgüzel, Ş.G., S. Rollas E.E. Oruç “Synthesis, Characterization and biological activity of novel 4-thiazolidinones and 1,3,4-oxadiazoles” 6th International Symposium on Pharmaceutical Sciences , Ankara-TURKEY, P-141, 27-29 June 2000.

15.

Küçükgüzel, İ., Ş.G.Küçükgüzel, S.Rollas “Some3-thioxo / alkylthio-1,2,4-triazoles with a substituted thiourea moiety as possible antimycobacterials.” 6th International Symposium on Pharmaceutical Sciences, Ankara-TURKEY, P-136, 27-29 June 2000.

16.

Küçükgüzel, Ş.G. and S.Rollas “ Synthesis, Characterization of Novel Coupling Products and 4-Arylhydrazono-2-pyrazoline-5-ones as Potential Antimycobacterial Agents” 3rd   International Symposium on Pharmaceutical Chemistry, İstanbul - TURKEY, Abstract P-23, 17-19 September 2001.

17.

Ş.G.Küçükgüzel, İ. Küçükgüzel, B.Oral, F.S.Sezen, S.Rollas “ HPLC-UV Diode Array and LC-MS/MS determination of in vivo metabolites of 4-nitro-2-phenoxymethansulfonanilide in rats” 1st International Meeting on Medicinal and Pharmaceutical Chemistry, Ankara - TURKEY, Abstract P65, 25-28 September 2002.

18.

Adil Mazi, Ş.Güniz Küçükgüzel, Fikrettin Şahin and Suzan Öztürk “Synthesis, characterization and antimicrobial activities of diflunisal hydrazide-hydrazones”1st International Meeting on Medicinal and Pharmaceutical Chemistry, Ankara - TURKEY, Abstract P66, 25-28 September 2002.

19.

Ş.Güniz Küçükgüzel, İlkay Küçükgüzel, Esra Tatar , Fikrettin Şahin, Medine Güllüce, Erik De Clercq “Synthesis of some novel heterocyclic compounds derived from diflunisal hydrazide as potential antimicrobial and antiviral agents ”2nd International Meeting on Medicinal and Pharmaceutical Chemistry, Antalya - TURKEY, P9, 10-14 October 2004.

20.

Ayla Kocatepe, Ş.Güniz Küçükgüzel, Erik De Clercq, Fikrettin Şahin, Medine Güllüce “New 4-thiazolidinones and related compounds : evaluation of antiviral , anti-HIV, antimycobacterial and antimicrobial activity” 2nd International Meeting on Medicinal and Pharmaceutical Chemistry, Antalya - TURKEY, P10, 10-14 October 2004.

21.

Koçyiğit-Kaymakçıoğlu, Oruç E.E., Yılmaz-Demircan F., Gürbüz Y., Kalaça S., Küçükgüzel Ş.G., Ülgen M., Rollas S. “A High Performance Liquid Chromatografic Method for the quantification of Cotinine in the ürine of preschool children” International Symposium  on Medicinal Chemistry Research and Development 2005, Kuşadası - TURKEY, P23, September 28-October 1, 2005.

22.

Küçükgüzel İ, Tatar E., Küçükgüzel Ş.G., Rollas S., De Clercq E., “Synthesis of Some novel thiourea derivatives obtained from 5-[(4-aminophenoxy)methyl]-4-methyl-2,4-dihydro-3H-1,2,4-triazole-3-thiones and evaluation as antiviral / anti-HIV agents” International Symposium  on Medicinal Chemistry Research and Development 2005, Kuşadası - TURKEY, P27, September 28-October 1, 2005.

23.

Neerja Kaushik-Basu, Alain Bopda-Waffo, Amartya Basu, Ye Chen, Tanaji T. Talele, Ş. Güniz Küçükgüzel4-Thiazolidinones: A Novel Class of Hepatitis C Virus NS5B Polymerase Inhibitors” XIXth International Symposium on Medicinal Chemistry , İstanbul , TURKEY. Abstract P-59. 29 August -2 September 2006 .

24.

Sevgi Karakuş, Ş.Güniz Küçükgüzel, İlkay Küçükgüzel, Erik De Clercq “Synthesis and antiviral activity of some novel thioureas derived from N-(4-nitro-2-phenoxyphenyl)-methanesulfonamide “XIXth International Symposium on Medicinal Chemistry , İstanbul , TURKEY. Abstract P-58. 29 August -2 September 2006 .

25.

Ş.Güniz Küçükgüzel, Pelin Çıkla, Sevim Rollas, İlkay Küçükgüzel, Erik De Clercq “Some novel thioureas derived from 4-aminobenzoic acid hydrazones as potential antiviral and antitubercular agents” XIXth International Symposium on Medicinal Chemistry , İstanbul , TURKEY. Abstract P-57. 29 August -2 September 2006 .

26.

F. Yılmaz-Demircan, E. Tatar , İ. Küçükgüzel, Ş.G.Küçükgüzel, E. De Clercq, F.Şahin, Ö.F.Bayrak “Synthesis and biological evaluation of some new 4-thiazolidinones as chemotherapeutic agents” XIXth International Symposium on Medicinal Chemistry , İstanbul , TURKEY. Abstract P-54. 29 August -2 September 2006 .

27.

Bedia Koçyiğit-Kaymakçıoğlu, Seda Ünsalan, Ş.Güniz Küçükgüzel, Göksel Şener, Sevim Rollas “HPLC-UV/DAD analysis for in vivo metabolites of 4-nitrobenzoic acid[(5-nitro-2-thiophenyl)methylene]hydrazide in rats” ” 6th AFMC International Medicinal Chemistry Symposıum, İstanbul , TURKEY. Abstract PB-79. 8 July -11 2007 .

28.

Esra Tatar, Pelin Çıkla, Ş.Güniz Küçükgüzel, İlkay Küçükgüzel, Fikrettin Şahin, Dilşad Yurdakul “ Synthesis and Biological activity of Flurbiprofen hydrazide derivatives” 5th   International Symposium on Pharmaceutical Chemistry, İstanbul - TURKEY, Abstract P-70, 5-7 September 2007.

 

Ulusal Kongreler

1.

Küçükgüzel, Ş.G.“Sübstitüe Arildiazonyum tuzlarının etilasetoasetat’la kenetlenme ürünleri ve bunlardan oluşan 2-pirazolin-5-on türevlerinin sentezi ve spektral verileri” M.Ü.Sağlık Bilimleri Enstitüsü-Doktora Günleri (Sözlü Bildiri), Doktora ve yüksek lisans tez özetleri, 35-40, İstanbul, 4 Kasım 1998.

2.

Ş.Güniz Küçükgüzel, Adil Mazi, Fikrettin Şahin , Suzan Öztürk ve James P.Stables “Diflunisal’den hareketle yeni hidrazit-hidrazonların sentezi ve yapılarının aydınlatılması” M.Ü.Sağlık Bilimleri Enstitüsü-Doktora Günleri (Poster), Doktora ve yüksek lisans tez özetleri, 129-130, İstanbul, 14 Kasım 2003.

3.

Ş.G.Küçükgüzel, İ. Küçükgüzel, B.Oral, F.S.Sezen, S.Rollas “ 4-Nitro-2-Fenoksimetansülfonanilid’in in vitro metabolizma çalışmasının HPLC-UV Diode Array (DAD) kullanarak Değerlendirilmesi” V.Ulusal Kromatografi Kongresi, 30 Haziran-2 Temmuz 2004, Özet Kitabı Sayfa no : 133.

4.

Sevgi Karakuş, İ. Küçükgüzel,  Ş.G.Küçükgüzel, “ Farmasötik Dozaj Formlarında Pseudoefedrin’in Setirizin ve Feksofenadin ile bir arada miktar tayini için yüksek basınçlı sıvı kromatografisi yönteminin geliştirilmesi ve validasyonu” V.Ulusal Kromatografi Kongresi, 30 Haziran-2 Temmuz 2004, Özet Kitabı Sayfa no : 91.

5.

Ayla Kocatepe, Ş.Güniz Küçükgüzel, Erik De Clercq, Fikrettin Şahin, Medine Güllüce “New 4-thiazolidinones and related compounds : evaluation of antiviral , anti-HIV, antimycobacterial and antimicrobial activity”. I.Ulusal Farmasötik Kimya Kongresi, İstanbul - TÜRKİYE, 11-12 Kasım 2006.

6.

Ayla Kocatepe, Ş.Güniz Küçükgüzel, Erik De Clercq, Fikrettin Şahin, Medine Güllüce “New 4-thiazolidinones and related compounds : evaluation of antiviral , anti-HIV, antimycobacterial and antimicrobial activity” T.C. Marmara Üniversitesi Sağlık Bilimleri Enstitüsü 8.Yüksek Lians ve Doktora Günleri, İstanbul - TÜRKİYE, 15 Haziran 2007.